Friday, January 6, 2012

PHARMACOLOGY


Receptor




Sympathetic
Major function
α1
↑ vascular smooth muscle contraction, ↑pupillary dilator muscle contraction (mydrasis), ↑ intestinal and bladder sphincter muscle contraction
α2
↓ sympathetic outflow, ↓ insulin release
β1
↑ heart rate, ↑ contractility, ↑ renin release, ↑ lipolysis
β2
Vasodilatation, bronchodilation, ↑ heart rate,
↑ contractility
↑ lipolysis, ↑ insulin release, ↓ uterine tone
M1



Parasympathetic
CNS, enteric nervous system
M2
↓ heart rate and contractility of atria
M3
↑ exocrine gland secretions, ↑ gut peristalsis, ↑ bladder contraction, bronchoconstriction, ↑ pupillary sphincter muscle contraction (miosis), ciliary muscle contraction (accommodation)
D1
Dopamine
Relaxes renal vascular smooth muscle
D2
Modulates transmitter release, especially in brain
H1

Histamine
↑ nasal and bronchial mucus production, contraction of bronchioles, pruritus, and pain
H2
↑ gastric acid secretion
V1
Vasopressin
↑ vascular smooth muscle contraction
V2
↑ H₂O permeability and reabsorption in the collecting tubule of the kidney (V2 is found in the 2 kidneys)


fuente: Le, Bhushan & Grimm 2011, First AID for the USMLE step 1

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